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ultiple neurochemical pathways are involved in
the pathology of Alzheimers disease (AD). The follow-
ing factors have been implicated in the development of
AD:
b
-amyloid; tau proteins; apolipoprotein E (APOE);
degeneration of cholinergic, serotonergic, and dopamin-
ergic neurons; oxidative damage; inflammation; estrogen
deficiency; and glutamatergic neurotransmission.
Neurochemical pathways for AD
b
-Amyloid
It has been suggested that deposits of
b
-amyloid proteins
appear to be the earliest morphological changes in the
formation of neuritic plaques.
1,2
These plaques ultimately
lead to the death and destruction of surrounding axons
and dendrites.
Tau proteins
Tau proteins are highly phosphorylated microtuble pro-
teins that form neurofibrillary tangles. These abnormal
filaments form either parallel bundles or randomly
arranged paired helical filaments that extend to the den-
dritic processes.
2
These tangles lead to dysfunction and
degeneration of nerve cells.
Apolipoprotein E
APOE is a cholesterol transport protein that has been
linked to late-onset familial and sporadic AD.
1-4
The gene
for this protein is found on chromosome 19 and is inher-
F r e e p a p e r
2 9 9
Combination pharmacotherapy in
Alzheimers disease
Jacobo Mintzer, MD; Dena Armstrong, MD; Warachal E. Faison, MD
M
Keywords:
Alzheimers disease; neurochemical pathway; combination therapy;
donezepil;
Gingko biloba
; NSAID; memantine; adverse effect
Author affiliations:
Ralph H. Johnson Veterans Administration Medical
Center, Charleston, SC, USA (Jacobo Mintzer); Alzheimers Research and Clinical Programs, Medical University of South Carolina, Charleston, SC, USA (Jacobo Mintzer, Dena Armstrong, Warachal E. Faison)
Address for correspondence:
Jacobo Mintzer, MD, Ralph H. Johnson
Veterans Administration Medical Center, Charleston, SC 29406, USA (e-mail: mintzerj@musc.edu)
This article is published following the 14th Biological Interface
Conference held in Rouffach, France, between October 1 and 5, 2002, on
the theme of Drug Development. Other articles from this meeting can
be found in
Dialogues in Clinical Neuroscience
(2002, Vol 4, No 4).
Alzheimers disease is a progressive, debilitating form of
dementia affecting more than 18 million people worldwide.
Without a cure, many patients and their families must turn
to long-term care institutions during the later stages of the
disease. Our current treatments only delay progression and
help control behavioral symptoms. In recent years, research
within this field has expanded to include many clinical trials
on potential drug therapies. However, despite the numer-
ous studies, the enigma of this disease remains. It is difficult,
yet necessary, to stay abreast of emerging information that
may warrant changes in current therapy. Rationale for com-
bination therapy becomes evident as we review the multi-
ple neurochemical pathways common to the disease. This
paper will review available information on Alzheimers dis-
ease pharmacotherapy, and evaluate data on the use of
combination drug therapy. Individual efficacy, possible syn-
ergistic effects, and the safety of combination therapy will
also be addressed.
© 2003, LLS SAS
Dialogues Clin Neurosci
. 2003;5:299-305.
Copyright © 2003 LLS SAS. All rights reserved
www.dialogues-cns.org